Other Name(s): P21, Waf1, P21
Assay:Inhibitory concentration against human p21 deficient cell (p21-/-) proliferation
Type:IC50
SMILES:COc1ccc(-c2nc(O)c3c4c(sc3n2)CCCC4)cc1OC
Value:>20000nM
Source:Homo sapiens
Assay:Inhibitory concentration against human p21 proficient cell (p21+/+) proliferation
Type:IC50
SMILES:COc1ccc(-c2nc(O)c3c4c(sc3n2)CCCC4)cc1OC
Value:>20000nM
Source:Homo sapiens
Assay:Inhibitory concentration against human p21 deficient cell (p21+/+) proliferation
Type:IC50
SMILES:COc1cc(-c2nc(O)c3c4c(sc3n2)CCCC4)cc(OC)c1OC
Value:>20000nM
Source:Homo sapiens
Assay:Inhibitory concentration against human p21 deficient cell (p21+/+) proliferation
Type:IC50
SMILES:O=C(c1cccs1)c1cnn2c(-c3cccc(NC(=O)C4CC4)c3)ccnc12
Value:=12000nM
Source:Homo sapiens
Assay:Inhibitory concentration against p21 deficient cell (p21-/-) proliferation
Type:IC50
SMILES:COC(=O)c1ccc(-c2nc(O)c3c4c(sc3n2)CCCC4)cc1
Value:>20000nM
Source:Homo sapiens
Assay:Inhibitory concentration against p21 deficient cell (p21-/-) proliferation
Type:IC50
SMILES:Oc1nc(-c2ccc(-c3ccccc3)cc2)nc2sc3c(c12)CCCC3
Value:>20000nM
Source:Homo sapiens
Assay:Inhibitory concentration against p21 deficient cell (p21-/-) proliferation
Type:IC50
SMILES:COc1cc(-c2nc(O)c3c4c(sc3n2)CCCC4)cc(OC)c1OC
Value:=2300nM
Source:Homo sapiens
Assay:Inhibitory concentration against p21 deficient cell (p21-/-) proliferation
Type:IC50
SMILES:Cc1ccc(-c2nc(O)c3c4c(sc3n2)CCCC4)cc1
Value:>20000nM
Source:Homo sapiens
Assay:Inhibitory concentration against p21 deficient cell (p21-/-) proliferation
Type:IC50
SMILES:COc1ccc(-c2nc(O)c3c4c(sc3n2)CCC4)cc1
Value:=2400nM
Source:Homo sapiens
Assay:Inhibitory concentration against p21 deficient cell (p21-/-) proliferation
Type:IC50
SMILES:COc1cc(OC)cc(-c2nc(O)c3c4c(sc3n2)CCCC4)c1
Value:>20000nM
Source:Homo sapiens
Assay:Inhibitory concentration against p21 deficient cell (p21-/-) proliferation
Type:IC50
SMILES:COc1ccc(-c2nc(O)c3c4c(sc3n2)CCCC4)cc1
Value:=2400nM
Source:Homo sapiens
Assay:Inhibitory concentration against p21 deficient cell (p21-/-) proliferation
Type:IC50
SMILES:CCOc1ccc(-c2nc(O)c3c4c(sc3n2)CCCC4)cc1
Value:=8400nM
Source:Homo sapiens
Assay:Inhibitory concentration against p21 deficient cell (p21-/-) proliferation
Type:IC50
SMILES:O=C(c1cccs1)c1cnn2c(-c3cccc(NC(=O)C4CC4)c3)ccnc12
Value:=400nM
Source:Homo sapiens
Assay:Inhibitory concentration against p21 deficient cell (p21-/-) proliferation
Type:IC50
SMILES:Oc1nc(-c2ccc(Cl)cc2)nc2sc3c(c12)CCCC3
Value:>20000nM
Source:Homo sapiens
Assay:Inhibitory concentration against p21 deficient cell (p21-/-) proliferation
Type:IC50
SMILES:COc1cc(-c2nc(O)c3ccsc3n2)cc(OC)c1OC
Value:>20000nM
Source:Homo sapiens
Assay:Inhibitory concentration against p21 deficient cell (p21-/-) proliferation
Type:IC50
SMILES:CCN(CC)c1ccc(-c2nc(O)c3c4c(sc3n2)CCCC4)cc1
Value:>20000nM
Source:Homo sapiens
Assay:Inhibitory concentration against p21 deficient cell (p21-/-) proliferation
Type:IC50
SMILES:COc1cc(-c2nc(O)c3c4c(sc3n2)CCC4)cc(OC)c1OC
Value:=3500nM
Source:Homo sapiens
Assay:Inhibitory concentration against p21 deficient cell (p21-/-) proliferation
Type:IC50
SMILES:COc1ccc(-c2nc(O)c3sccc3n2)cc1
Value:>20000nM
Source:Homo sapiens
Assay:Inhibitory concentration against p21 deficient cell (p21-/-) proliferation
Type:IC50
SMILES:COc1cc(-c2nc(O)c3sccc3n2)cc(OC)c1OC
Value:>20000nM
Source:Homo sapiens
Assay:Inhibitory concentration against p21 deficient cell (p21-/-) proliferation
Type:IC50
SMILES:O=[N+]([O-])c1ccc(-c2nc(O)c3c4c(sc3n2)CCCC4)cc1
Value:>20000nM
Source:Homo sapiens

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