Assay: Inhibition of Insulin receptor kinase-beta Type: IC50 SMILES: CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4c(c5c6ccccc6n2c5c31)C(=O)NC4 Value: =200nM Source:
	Assay: Inhibition of Insulin receptor kinase-beta Type: IC50 SMILES: CCN1CCOCCn2cc(c3ccccc32)C2=C(C(=O)NC2=O)c2cn(c3ccccc23)CCOCC1 Value: >100000nM Source:
	Assay: Concentration required to achieve 50% inhibition of tyrosine phosphorylation on human Insulin-like growth factor I receptor Type: IC50 SMILES: CC(C)c1cc(/C=C2\C(=O)Nc3ccccc32)cc(C(C)C)c1O Value: =10100nM Source:
	Assay: Concentration required to achieve 50% inhibition of tyrosine phosphorylation on human Insulin-like growth factor I receptor Type: IC50 SMILES: Cc1cccc2c1/C(=C/c1ccc[nH]1)C(=O)N2 Value: >100000nM Source:
	Assay: Concentration required to achieve 50% inhibition of tyrosine phosphorylation on human Insulin-like growth factor I receptor Type: IC50 SMILES: O=C1Nc2ccccc2/C1=C/c1ccc[nH]1 Value: >100000nM Source:
	Assay: Concentration required to achieve 50% inhibition of tyrosine phosphorylation on human Insulin-like growth factor I receptor Type: IC50 SMILES: CCOC(=O)c1c(C)[nH]c(/C=C2\C(=O)Nc3ccccc32)c1C Value: >100000nM Source:
	Assay: Concentration required to achieve 50% inhibition of tyrosine phosphorylation on human Insulin-like growth factor I receptor Type: IC50 SMILES: O=C1Nc2ccc(Br)cc2/C1=C/c1ccc(N2CCOCC2)cc1 Value: >10000nM Source:
	Assay: Concentration required to achieve 50% inhibition of tyrosine phosphorylation on human Insulin-like growth factor I receptor Type: IC50 SMILES: COc1ccc(/C=C2\C(=O)Nc3ccccc32)cc1C(C)(C)C Value: >100000nM Source:
	Assay: Concentration required to achieve 50% inhibition of tyrosine phosphorylation on human Insulin-like growth factor I receptor Type: IC50 SMILES: Cc1c[nH]c(/C=C2\C(=O)Nc3ccccc32)c1CCC(=O)O Value: >100000nM Source:
	Assay: Concentration required to achieve 50% inhibition of tyrosine phosphorylation on human Insulin-like growth factor I receptor Type: IC50 SMILES: O=C1Nc2cc(F)ccc2/C1=C/c1ccc[nH]1 Value: >100000nM Source:
	Assay: Concentration required to achieve 50% inhibition of tyrosine phosphorylation on human Insulin-like growth factor I receptor Type: IC50 SMILES: O=C1Nc2ccccc2/C1=C/c1n[nH]cc1Cl Value: >100000nM Source:
	Assay: Concentration required to achieve 50% inhibition of tyrosine phosphorylation on human Insulin-like growth factor I receptor Type: IC50 SMILES: O=C1Nc2ccccc2/C1=C/c1ccc(Br)cc1 Value: >100000nM Source:
	Assay: Concentration required to achieve 50% inhibition of tyrosine phosphorylation on human Insulin-like growth factor I receptor Type: IC50 SMILES: CCc1ccc(/C=C2/C(=O)Nc3ccccc32)o1 Value: >100000nM Source:
	Assay: Concentration required to achieve 50% inhibition of tyrosine phosphorylation on human Insulin-like growth factor I receptor Type: IC50 SMILES: Cc1cccc2c1/C(=C/c1ccc(N3CCN(C=O)CC3)cc1)C(=O)N2 Value: =67600nM Source:
	Assay: Concentration required to achieve 50% inhibition of tyrosine phosphorylation on human Insulin-like growth factor I receptor Type: IC50 SMILES: CSc1ccc(/C=C2\C(=O)Nc3cccc(C)c32)s1 Value: >100000nM Source:
	Assay: Concentration required to achieve 50% inhibition of tyrosine phosphorylation on human Insulin-like growth factor I receptor Type: IC50 SMILES: Cc1cccc2c1/C(=C/c1ccc(N3CCOCC3)cc1)C(=O)N2 Value: >100000nM Source:
	Assay: Concentration required to achieve 50% inhibition of tyrosine phosphorylation on human Insulin-like growth factor I receptor Type: IC50 SMILES: CC(C)c1cc(/C=C2\C(=O)Nc3ccc(Cl)cc32)cc(C(C)C)c1O Value: >100000nM Source:
	Assay: Concentration required to achieve 50% inhibition of tyrosine phosphorylation on human Insulin-like growth factor I receptor Type: IC50 SMILES: O=C1Nc2ccccc2/C1=C/c1ccc(N2CCOCC2)cc1 Value: >100000nM Source:
	Assay: Concentration required to achieve 50% inhibition of tyrosine phosphorylation on human Insulin-like growth factor I receptor Type: IC50 SMILES: O=C1Nc2ccccc2/C1=C/c1ccc(N2CCCC2)cc1 Value: >100000nM Source:
	Assay: Concentration required to achieve 50% inhibition of tyrosine phosphorylation on human Insulin-like growth factor I receptor Type: IC50 SMILES: COc1c(Br)cc(/C=C2\C(=O)Nc3ccccc32)cc1C(C)(C)C Value: >100000nM Source:

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